Trifluoperazine N-Glucuronide
Based on 1 Customer Validation
Trifluoperazine N-Glucuronide (UGT1A4), as one of the human UGT1A isoforms, is expressed in the liver. Trifluoperazine N-Glucuronide catalyzes the imipramine and trifluoperazine Nglucuronide formation.
For research use only. We do not sell to patients.
- Purity: 95.80%
- CAS No.: 165602-90-4
- Formula: C27H32F3N3O6S
- Molecular Weight:583.62
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Storage:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
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Biological Activity
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Chemical Information
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Solvent & Solubility
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Trifluoperazine N-Glucuronide (1~10 μg; HEK293 cells) expression levels is 0.14 unit/mg protein[1].
Trifluoperazine N-Glucuronide coexpression affects the activity of human UGT1A9. The imipramine N-glucuronide formation by the single expression system of trifluoperazine N-Glucuronide follows the Michaelis-Menten equation. Trifluoperazine N-Glucuronide interacts with the human UGT1A1 and UGT1A6, affecting the enzymatic activities[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 165602-90-4
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Appearance Solid
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Molecular Weight 583.62
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Formula C27H32F3N3O6S
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Color Off-white to light yellow
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SMILES
FC(C(C=C1N2CCCN3CC[N+](C)([C@H]4[C@@H]([C@H]([C@@H]([C@@H](C([O-])=O)O4)O)O)O)CC3)=CC=C1SC5=C2C=CC=C5)(F)F
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Synonyms
UGT1A4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 25 mg/mL (42.84 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (273 KB)
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SDS (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.7134 mL | 8.5672 mL | 17.1344 mL | 42.8361 mL |
| 5 mM | 0.3427 mL | 1.7134 mL | 3.4269 mL | 8.5672 mL | |
| 10 mM | 0.1713 mL | 0.8567 mL | 1.7134 mL | 4.2836 mL | |
| 15 mM | 0.1142 mL | 0.5711 mL | 1.1423 mL | 2.8557 mL | |
| 20 mM | 0.0857 mL | 0.4284 mL | 0.8567 mL | 2.1418 mL | |
| 25 mM | 0.0685 mL | 0.3427 mL | 0.6854 mL | 1.7134 mL | |
| 30 mM | 0.0571 mL | 0.2856 mL | 0.5711 mL | 1.4279 mL | |
| 40 mM | 0.0428 mL | 0.2142 mL | 0.4284 mL | 1.0709 mL |
Trifluoperazine N-Glucuronide Related Classifications
HY-137083 Related Classifications
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