2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor
  4. Trimazosin

Trimazosin is an orally active, quinazoline derivative which is structurally related to prazosin. Trimazosin shows hypotensive effect by selectively block α1-adrenoceptors.

For research use only. We do not sell to patients.

Trimazosin Chemical Structure

Trimazosin Chemical Structure

CAS No. : 35795-16-5

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Trimazosin Related Antibodies

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Description

Trimazosin is an orally active, quinazoline derivative which is structurally related to prazosin. Trimazosin shows hypotensive effect by selectively block α1-adrenoceptors[1][2].

IC50 & Target

α1-adrenergic receptor

 

In Vivo

Trimazosin (10–30 mg/kg; i.h.; once) produces graded decreases in blood pressure[3].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Conscious spontaneously hypertensive rats (SHR)[3]
Dosage: 10–30 mg/kg
Administration: Subcutaneous administration, once
Result: Produced graded decreases in blood pressure.
Molecular Weight

435.47

Formula

C20H29N5O6
CAS No.
SMILES

O=C(N1CCN(CC1)C2=NC3=C(C=C(C(OC)=C3OC)OC)C(N)=N2)OCC(C)(C)O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Trimazosin Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Trimazosin35795-16-5Adrenergic ReceptorBeta ReceptorQuinazoline derivativePrazosinHypotensive effectInhibitorinhibitorinhibit

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