VL-0395
VL-0395 is a CCK1 selective antagonist with IC50 of 0.197 μM for CCK1 in rat pancreatic acinar cells.
For research use only. We do not sell to patients.
- CAS No.: 620167-11-5
- Formula: C25H21N3O4
- Molecular Weight:427.45
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| A-431 | IC50 |
197 nM
Compound: VL-0395
|
Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor in A431 cells
Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor in A431 cells
|
[PMID: 16610788] |
Chemical Information
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CAS No. 620167-11-5
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Molecular Weight 427.45
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Formula C25H21N3O4
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SMILES
O=C(C(CC1=CC=CC=C1)NC(C2=C(NC(C3=CC4=C(N3)C=CC=C4)=O)C=CC=C2)=O)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)