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β2AR ligand 1

β2AR ligand 1 (Compound 4) is a homobivalent bitopic ligand for β2 adrenergic receptor (β2AR) on the orthosteric binding site (OBS) and the metastable binding sites (MBS).

For research use only. We do not sell to patients.

CAS No.: 3051498-44-0
Formula: C₃₃H₄₉N₅O₄
Molecular Weight:579.77

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (263 KB)

β2AR ligand 1 Chemical Structure

CAS No.: 3051498-44-0

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Sample (0.1mg)

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(In Japan)

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

β2AR ligand 1 (Compound 4) is a homobivalent bitopic ligand for β2 adrenergic receptor (β2AR) on the orthosteric binding site (OBS) and the metastable binding sites (MBS)^[1].

All Adrenergic Receptor Isoforms :

Chemical Information

CAS No. 3051498-44-0
Molecular Weight 579.77
Formula C₃₃H₄₉N₅O₄
SMILES

C=CCC1=C(C=CC=C1)OC[C@H](CNCCCC2=CN(N=N2)CCCCC3=CC=C(C=C3)OC[C@H](CNC(C)C)O)O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (263 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Gaiser BI, et al., Bitopic Ligands Support the Presence of a Metastable Binding Site at the β2 Adrenergic Receptor. J Med Chem. 2024 Jul 11;67(13):11053-11068. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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