[Des-Arg9]-Bradykinin
Based on 2 publication(s) in Google Scholar
[Des-Arg9]-Bradykinin is a Bradykinin (B1) receptor agonist that displays selectivity for B1 over B2 receptors.
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- CAS No.: 15958-92-6
- Formule: C44H61N11O10
- Masse moléculaire:904.02
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications Citing Use of MedChemExpress (MCE) [Des-Arg9]-Bradykinin
MoreVoir tous les produits spécifiques à Isoform Bradykinin Receptor
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Activité biologique
Description
IC50 & Target
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Bradykinin B1 Receptor (B1R) |
In Vitro
The B2 receptor mediates the action of bradykinin (BK) and lysyl-bradykinin (Lys-BK), the first set of bioactive kinins formed in response to injury from kininogen precursors through the actions of plasma and tissue kallikreins, whereas the B1 receptor mediates the action of [Des-Arg9]-Bradykinin (des-Arg9-BK) and Lys-des-Arg Arg9-BK, the second set of bioactive kinins formed through the actions of carboxypeptidases on BK and Lys-BK, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 15958-92-6
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Masse moléculaire 904.02
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Formule C44H61N11O10
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Sequence
Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe
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Sequence Shortening
RPPGFSPF
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications (2)
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Journal Impact Factor
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Most Recent
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Nat Commun
Endothelial Sp1/Sp3 are essential to the effect of captopril on blood pressure in male mice. [Abstract]2023 Sep 21;14(1):5891. PMID: 37735515 -
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)