1. GPCR/G Protein Neuronal Signaling
  2. 5-HT Receptor
  3. 5-HT6/5-HT2AR antagonist-1

5-HT6/5-HT2AR antagonist-1 is a potent dual 5-HT6/5-HT2AR antagonist with Ki values of 11 nM and 39 nM, respectively.

For research use only. We do not sell to patients.

5-HT6/5-HT2AR antagonist-1 Chemical Structure

5-HT6/5-HT2AR antagonist-1 Chemical Structure

CAS No. : 2763654-60-8

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Description

5-HT6/5-HT2AR antagonist-1 is a potent dual 5-HT6/5-HT2AR antagonist with Ki values of 11 nM and 39 nM, respectively[1].

IC50 & Target[1]

5-HT2A Receptor

39 nM (Ki)

5-HT6 Receptor

11 nM (Ki)

Molecular Weight

394.54

Formula

C21H26N6S

CAS No.
SMILES

NC1=NC(N2CCN(C)CC2)=NC(C(C)(SC3=CC=C4C=CC=CC4=C3)C)=N1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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5-HT6/5-HT2AR antagonist-1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
5-HT6/5-HT2AR antagonist-1
Cat. No.:
HY-145862
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