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Cat. No.: HY-101683

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Deriglidole

Name: Deriglidole
Brand: MedChemExpress
SKU: HY-101683
Price: 753.00 USD
Availability: InStock
Rating: 5 (1 reviews)

(Synonyms: SL 86-0715)

Deriglidole is a peripheral adrenoceptor antagonist with a high affinity for α₂-adrenoceptors.

For research use only. We do not sell to patients.

CAS No.: 122830-14-2
Formula: C₁₆H₂₁N₃
Molecular Weight:255.36

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (273 KB)

Deriglidole Chemical Structure

CAS No.: 122830-14-2

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
- In Vitro
Chemical Information
Purity & Documentation
References
Calculators
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Biological Activity

Description

Deriglidole is a peripheral adrenoceptor antagonist with a high affinity for α₂-adrenoceptors.

IC₅₀ & Target

Adrenoceptor^[1]

All Adrenergic Receptor Isoforms :

In Vitro

Deriglidole is a selective α₂-receptor inhibitor. Deriglidole inhibits [³H]Clonidine and [³H]Idazoxan but not [³H]Prazosin binding to rat cortical and human platelet α₂-adrenoceptors and is more selective than Idazoxan for peripheral receptors^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 122830-14-2
Molecular Weight 255.36
Formula C₁₆H₂₁N₃
SMILES

CCCC1(C2=NCCN2)N3C4=C(C=CC=C4CC3)C1
Synonyms

SL 86-0715
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (273 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Natali A, et al. Effects of acute alpha 2-blockade on insulin action and secretion in humans. Am J Physiol. 1998 Jan;274(1 Pt 1):E57-64. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Biological Activity
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- IC₅₀ & Target
- In Vitro
Chemical Information
Purity & Documentation
References

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Deriglidole

All Adrenergic Receptor Isoforms