1. PROTAC
  2. Ligand for E3 Ligase
  3. E3 ligase Ligand 9

E3 ligase Ligand 9 

Cat. No.: HY-122725 Purity: 98.94%
Handling Instructions

E3 ligase Ligand 9 is a Ligand of BETd-260 for E3 Ligase used in PROTAC. BETd-260 is a potent BET degrader based on PROTAC technology, with an IC50 of 51 pM against BRD4 protein in RS4;11 leukemia cell line.

For research use only. We do not sell to patients.

E3 ligase Ligand 9 Chemical Structure

E3 ligase Ligand 9 Chemical Structure

CAS No. : 2093388-45-3

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 440 In-stock
Estimated Time of Arrival: December 31
100 mg USD 400 In-stock
Estimated Time of Arrival: December 31
500 mg USD 950 In-stock
Estimated Time of Arrival: December 31
1 g USD 1600 In-stock
Estimated Time of Arrival: December 31
2 g USD 2600 In-stock
Estimated Time of Arrival: December 31
5 g   Get quote  
10 g   Get quote  

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Based on 1 publication(s) in Google Scholar

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  • Biological Activity

  • Technical Information

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  • References

Description

E3 ligase Ligand 9 is a Ligand of BETd-260 for E3 Ligase used in PROTAC. BETd-260 is a potent BET degrader based on PROTAC technology, with an IC50 of 51 pM against BRD4 protein in RS4;11 leukemia cell line[1].

IC50 & Target

E3 ligase[1].

Storage

-20°C, stored under nitrogen

References
Molecular Weight

329.39

Formula

C₁₈H₂₃N₃O₃

CAS No.

2093388-45-3

SMILES

O=C(C(N(CC1=C2C=CC=C1CCCCCN)C2=O)CC3)NC3=O

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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C1   V1   C2   V2

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Product Name:
E3 ligase Ligand 9
Cat. No.:
HY-122725
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E3 ligase Ligand 9

Cat. No.: HY-122725