1. Metabolic Enzyme/Protease
  2. Fatty Acid Synthase (FASN)
  3. HS79

HS79 

Cat. No.: HY-112522
Handling Instructions

HS-79 is an enantiomer of Fasnall, which is a selective fatty acid synthase (FASN) inhibitor. HS-79 is able to inhibit the incorporation of tritiated acetate into lipids with an IC50 of 1.57 μM.

For research use only. We do not sell to patients.

HS79 Chemical Structure

HS79 Chemical Structure

CAS No. : 2138838-56-7

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Description

HS-79 is an enantiomer of Fasnall, which is a selective fatty acid synthase (FASN) inhibitor. HS-79 is able to inhibit the incorporation of tritiated acetate into lipids with an IC50 of 1.57 μM.

IC50 & Target

FASN[1]

In Vitro

Fasnall, a thiophenopyrimidine selectively targeting FASN through its co-factor binding sites. Fasnall has anti-proliferative activity and induces apoptosis in breast cancer cells[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

338.47

Formula

C₁₉H₂₂N₄S

CAS No.

2138838-56-7

SMILES

CC1=C(C)SC2=NC=NC(N[[email protected]@H]3CCN(CC4=CC=CC=C4)C3)=C21

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

HS79HS 79HS-79Fatty Acid Synthase (FASN)Inhibitorinhibitorinhibit

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HS79
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