1. Metabolic Enzyme/Protease
  2. MAGL
  3. PF-06795071

PF-06795071 

Cat. No.: HY-111512
Handling Instructions

PF-06795071 is a potent and selective covalent MAGL inhibitor with an IC50 of 3 nM.

For research use only. We do not sell to patients.

PF-06795071 Chemical Structure

PF-06795071 Chemical Structure

CAS No. : 2075629-81-9

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Description

PF-06795071 is a potent and selective covalent MAGL inhibitor with an IC50 of 3 nM[1].

IC50 & Target

IC50: 3 nM (MAGL)[1]

In Vitro

PF-06795071 shows excellent selectivity against FAAH with an IC50 of 3.1 μM[1].

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

399.34

Formula

C₁₈H₁₇F₄N₃O₃

CAS No.

2075629-81-9

SMILES

OC[[email protected]](C(F)(F)F)OC(N1C[[email protected]]([[email protected]@]2([H])C1)([H])[[email protected]]2C3=NN(C4=CC=C(F)C=C4)C=C3)=O

Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
PF-06795071
Cat. No.:
HY-111512
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PF-06795071

Cat. No.: HY-111512