AG-041R
Based on 1 Customer Validation
AG-041R is a potent and selective CCK2 Receptor/Gastrin antagonist. AG-041R inhibits gastrin-evoked secretion of pancreastatin with an IC50 of 2.2 nM. AG-041R inhibits cell growth of Mastomys ECL carcinoid tumor cells.
For research use only. We do not sell to patients.
- Purity: 99.9%
- CAS No.: 159883-95-1
- Formula: C31H36N4O5
- Molecular Weight:544.64
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Storage:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Chemical Information
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CAS No. 159883-95-1
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Appearance Solid
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Molecular Weight 544.64
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Formula C31H36N4O5
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Color White to off-white
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SMILES
CC(C=C1)=CC=C1NC(C[C@]2(C3=CC=CC=C3N(C2=O)CC(OCC)OCC)NC(NC4=CC=C(C=C4)C)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Purity & Documentation
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Data Sheet (273 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
[1]. Ding XQ, et al. Evaluation of three novel cholecystokinin-B/gastrin receptor antagonists: a study of their effects on rat stomach enterochromaffin-like cell activity. Pharmacol Toxicol. 1997 Nov;81(5):232-7. [Content Brief]
[2]. Lindström, E., et al. Pharmacological analysis of CCK2 receptor antagonists using isolated rat stomach ECL cells. Br. J. Pharmacol. 127(2), 530-536 (1999). [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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