Aplithianines A
Aplithianines A is a potent inhibitor against J-PKAcα with an IC50 of 1 μM , and inhibits wild-type PKA with an IC50 of 84 nM. Aplithianines A inhibits J-PKAcα catalytic activity by competitively binding to the ATP pocket.
For research use only. We do not sell to patients.
- CAS No.: 3027425-38-0
- Formula: C13H13N7S
- Molecular Weight:299.35
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
1 μM (J-PKAcα)[1]
Chemical Information
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CAS No. 3027425-38-0
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Molecular Weight 299.35
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Formula C13H13N7S
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SMILES
CN1C=NC=C1C(SCC2)=CN2C3=NC=NC4=C3N=CN4
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Structure Classification
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Initial Source
Aplidium sp.
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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