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Art. -Nr.: HY-182715

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PSB-10211

PSB-10211 is a P2X2 receptor antagonist with an IC₅₀ of 0.086 μM against rat P2X2 receptors. PSB-10211 inhibits ATP-mediated currents of rat P2X2 receptors expressed in Xenopus oocytes. PSB-10211 can be used in studies related to pain and urinary incontinence.

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CAS. Nr.: 66295-57-6
Formel: C₂₃H₁₃Cl₂N₆NaO₅S
Molecular Weight:579.35

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Please store the product under the recommended conditions in the Certificate of Analysis.

PSB-10211 Chemical Structure

CAS. Nr.: 66295-57-6

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Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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Biologische Aktivität

Beschreibung

Alle P2X Receptor Isoform-spezifische Produkte anzeigen :

In Vitro

PSB-10211 inhibits human P2Y₂ receptor-mediated calcium mobilization with an IC₅₀ of 24.3 μM, shows inhibitory activity with an IC₅₀ of ~10 μM at human P2Y₄ receptors, and shows inhibitory activity at concentrations >10 μM at rat P2Y₆ receptors^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS. Nr. 66295-57-6
Molecular Weight 579.35
Formel C₂₃H₁₃Cl₂N₆NaO₅S
SMILES

O=C1C2=C(C(C3=C(C(S(=O)(O[Na])=O)=CC(NC4=CC(NC5=NC(Cl)=NC(Cl)=N5)=CC=C4)=C13)N)=O)C=CC=C2
Versand

Room temperature in continental US; may vary elsewhere.
Speicherung

Please store the product under the recommended conditions in the Certificate of Analysis.

Reinheit & Dokumentation

Handling Instructions (2659 KB)

Verweise

[1]. Baqi Y, et al. Discovery of potent competitive antagonists and positive modulators of the P2X2 receptor. J Med Chem. 2011;54(3):817-830. [Content Brief]

Calculators

Molaritätsrechner

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Konzentration Konzentration

Volumen Volumen

Molecular Weight Molecular Weight

Verdünnungsrechner

Konzentration _{(Stammlösung)} × Volumen _{(Stammlösung)} = Konzentration _{(Ziellösung)} × Volumen _{(Ziellösung)}

Konzentration _{(Stammlösung)} Konzentration _{(Stammlösung)}

Volumen _{(Stammlösung)} Volumen _{(Stammlösung)}

Konzentration _{(Ziellösung)} Konzentration _{(Ziellösung)}

Volumen _{(Ziellösung)} Volumen _{(Ziellösung)}

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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PSB-10211

High-Throughput Bioactive Compound Library

Alle P2X Receptor Isoform-spezifische Produkte anzeigen

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PSB-10211 Related Classifications

HY-182715 Related Classifications