AR-M1896
AR-M1896 is a GalR2 selective agonist with a binding IC50 of 1.76 nM for rat GalR2. AR-M1896 can be used for the research of acute myocardial infarction and neuropathic pain.
Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.
- CAS No.: 367518-31-8
- Formule: C54H81N13O14
- Masse moléculaire:1136.30
-
Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Voir tous les produits spécifiques à Isoform Neuropeptide Y Receptor
More
Activité biologique
IC50: 1.76 nM (rat GalR2), 879 nM (hGalR1)[1]
Chemical Information
-
CAS No. 367518-31-8
-
Masse moléculaire 1136.30
-
Formule C54H81N13O14
-
Sequence
Trp-Thr-Leu-Asn-Ser-Ala-Gly-Tyr-Leu-Leu-NH2
-
Sequence Shortening
WTLNSAGYLL-NH2
-
Livraison
Room temperature in continental US; may vary elsewhere.
-
Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
[1]. Liu HX, et al. Receptor subtype-specific pronociceptive and analgesic actions of galanin in the spinal cord: selective actions via GalR1 and GalR2 receptors. Proc Natl Acad Sci U S A. 2001 Aug 14;98(17):9960-4. [Content Brief]
[2]. Serebryakova L, et al. Galanin and its N-terminal fragments reduce acute myocardial infarction in rats. Peptides. 2019 Jan;111:127-131. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)