AY254
AY254 is an analogue of AY77 (HY-138951). AY254 is ERK-biased PAR2 agonist with an EC50 of 2 nM. AY254 relieves cytokine-induced caspase 3/8 activation. AY254 also promotes scratch-wound healing and induced IL-8 secretion via PAR2-ERK1/2 signaling
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- CAS No.: 2093408-03-6
- Formule: C30H49N9O6
- Masse moléculaire:631.77
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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PAR2 2 nM (EC50) |
Chemical Information
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CAS No. 2093408-03-6
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Masse moléculaire 631.77
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Formule C30H49N9O6
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Sequence
{5-Isoxazolylcarbonyl-Cha}-{Chg}-Ala-Arg-NH2
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Sequence Shortening
{5-Isoxazolylcarbonyl-Cha}-{Chg}-AR-NH2
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)