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Cat. No.: HY-117379

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CHIR-2279

CHIR-2279 is a high-affinity ligand (K_i=5 nM) for the α₁-adrenergic receptor and can be further studied as a drug lead compound.

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CAS No.: 158198-45-9
Formule: C₃₄H₃₆N₄O₄
Masse moléculaire:564.67

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (266 KB)

CHIR-2279 Chemical Structure

CAS No.: 158198-45-9

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
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Activité biologique

Description

CHIR-2279 is a high-affinity ligand (K_i=5 nM) for the α₁-adrenergic receptor and can be further studied as a drug lead compound^[1].

IC₅₀ & Target^[1]

α1-adrenergic receptor

5 nM (Ki)

Voir tous les produits spécifiques à Isoform Adrenergic Receptor :

Chemical Information

CAS No. 158198-45-9
Masse moléculaire 564.67
Formule C₃₄H₃₆N₄O₄
SMILES

O=C(CN(CCC1=CC=CC=C1)C(CN(C(CNCCC2=CC=C(C=C2)O)=O)C3=CC=C(C4=CC=CC=C4)C=C3)=O)N
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (266 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Zuckermann, et al. Discovery of nanomolar ligands for 7-transmembrane G-protein-coupled receptors from a diverse N-(substituted) glycine peptoid library. Journal of medicinal chemistry 37.17 (1994): 2678-2685. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

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Concentration _(final) Concentration _(final)

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références

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CHIR-2279

Voir tous les produits spécifiques à Isoform Adrenergic Receptor

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

CHIR-2279 Related Classifications

HY-117379 Related Classifications