(E)-SI-2
(E)-SI-2 is an isomer of SI-2, an inhibitor of the steroid receptor coactivator SRC-3. SI-2 has anticancer activity and increases the number of cytotoxic immune cells in mice with breast cancer.
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- CAS No.: 380537-35-9
- Formule: C15H15N5
- Masse moléculaire:265.31
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
SRC-3[1]
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| TOV112D | EC50 |
0.004 μM
Compound: C9
|
Growth inhibition of human TOV112D cells harbouring p53 R175H mutant incubated for 3 days by MTS assay
Growth inhibition of human TOV112D cells harbouring p53 R175H mutant incubated for 3 days by MTS assay
|
[PMID: 33538587] |
Chemical Information
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CAS No. 380537-35-9
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Masse moléculaire 265.31
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Formule C15H15N5
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SMILES
CN1C2=CC=CC=C2N=C1N/N=C(C3=CC=CC=N3)\C
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Synonyms
(E)-EPH 116
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)