Giclanfentrine
Giclanfentrine is a potent PDE3A inhibitor with an IC50 of 0.0058 μM. Giclanfentrine inhibits PDE4B1 activity with an IC50 of 12.9 μM. Giclanfentrine is applicable to studies related to PDE3/cAMP signaling.
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- CAS No.: 2408152-69-0
- Formule: C30H35N7O5
- Masse moléculaire:573.64
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Help & FAQs
Activité biologique
Description
IC50 & Target
[1]|
PDE3A 0.0058 μM (IC50) |
PDE4B1 12.9 μM (IC50) |
In Vitro
Giclanfentrine (compound 23) inhibits the activities of recombinant PDE3A and PDE4B1 enzymes, with IC50 values of 0.0058 μM and 12.9 μM, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .
Chemical Information
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CAS No. 2408152-69-0
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Masse moléculaire 573.64
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Formule C30H35N7O5
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SMILES
O=C(C1=C(N=NN1C)O)NCCN2/C(C=C3C4=C(CCN3C2=O)C=C(OCC)C(OC)=C4)=N/C5=C(C)C=C(C)C=C5C
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Giclanfentrine Related Classifications
HY-171827 Related Classifications
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