MRS2802
MRS2802 is a P2Y14 receptor agonist with an EC50 value of 63 nM. MRS2802 can effectively activate the P2Y14 receptor and may play a role in regulating platelet function. The selectivity and activity of MRS2802 are conducive to in-depth research on the biological functions and pharmacological properties of P2Y receptors. The development of MRS2802 provides a potential inhibitory strategy for the search for new antiplatelet compounds.
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- CAS No.: 1047980-53-9
- Formule: C10H14F2N2O11P2
- Masse moléculaire:438.17
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Activité biologique
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HEK293 | EC50 |
63 nM
Compound: 12
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Agonist activity at human P2Y14 receptor expressed in HEK293 cells coexpressing phospholipase C-activating Gi protein cells assessed as inhibition of forskolin induced [3H]cAMP production
Agonist activity at human P2Y14 receptor expressed in HEK293 cells coexpressing phospholipase C-activating Gi protein cells assessed as inhibition of forskolin induced [3H]cAMP production
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[PMID: 19902968] |
Chemical Information
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CAS No. 1047980-53-9
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Masse moléculaire 438.17
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Formule C10H14F2N2O11P2
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SMILES
O=C(C=CN1[C@@H]2O[C@H](COP(O)(C(P(O)(O)=O)(F)F)=O)[C@@H](O)[C@H]2O)NC1=O
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
MRS2802 Related Classifications
HY-122211 Related Classifications
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