Carbazeran citrate
Carbazeran (citrate), a potent phosphodiesterase inhibitor, is aldehyde oxidase substrate. Carbazeran (citrate) can be used for the research of metabolic disease.
For research use only. We do not sell to patients.
- CAS No.: 153473-94-0
- Formula: C24H32N4O11
- Molecular Weight:552.53
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
phosphodiesterase[1]
Oral administration of carbazeran (citrate) to guinea pigs has reportedly resulted in large kinetic deuterium isotope effects on the AUC and Cmax, without a change of systemic half-life[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
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Animal Model:Mice[1]
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Dosage:10 mg/kg
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Administration:P.o.
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Result:The mean plasma concentrations were lower than in those from control mice for 0.5~4 hours after oral administration.
Chemical Information
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CAS No. 153473-94-0
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Molecular Weight 552.53
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Formula C24H32N4O11
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SMILES
O=C(OC1CCN(C2=NN=CC3=C2C=C(OC)C(OC)=C3)CC1)NCC.O=C(CC(C(O)=O)(O)CC(O)=O)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)