1449685-96-4
1449685-96-4
Chemical Structure
DDR1-IN-1
- CAS No.: 1449685-96-4
- Formula:C30H31F3N4O3
- Molecular Weight:552.59
IUPAC Name: 4-((4-ethylpiperazin-1-yl)methyl)-N-(4-methyl-3-((2-oxoindolin-5-yl)oxy)phenyl)-3-(trifluoromethyl)benzamide
InChIKey: AOZPVMOOEJAZGK-UHFFFAOYSA-N
SMILES: O=C(NC1=CC=C(C)C(OC2=CC3=C(NC(C3)=O)C=C2)=C1)C4=CC=C(CN5CCN(CC)CC5)C(C(F)(F)F)=C4
Biological Activity: DDR1-IN-1 is a potent and selective DDR1 receptor tyrosine kinase inhibitor with an IC50 of 105 nM; 4-fold less potent for DDR2 (IC50 = 413 nM)[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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DDR1-IN-1 | 98.0% | DDR1-IN-1 is a potent and selective DDR1 receptor tyrosine kinase inhibitor with an IC50 of 105 nM; 4-fold less potent for DDR2 (IC50 = 413 nM). | ||||||||||||||||||||
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References
Keywords
