199864-86-3
199864-86-3
Chemical Structure
RS-127445 hydrochloride
- CAS No.: 199864-86-3
- Formula:C17H17ClFN3
- Molecular Weight:317.79
IUPAC Name: 4-(4-fluoronaphthalen-1-yl)-6-isopropylpyrimidin-2-amine hydrochloride
InChIKey: MKJPYBJBPRFMHL-UHFFFAOYSA-N
SMILES: NC1=NC(C(C)C)=CC(C2=C3C=CC=CC3=C(F)C=C2)=N1.[H]Cl
Biological Activity: RS-127445 hydrochloride is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. RS-127445 hydrochloride shows 1000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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RS-127445 hydrochloride | 99.78% | RS-127445 hydrochloride is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. RS-127445 hydrochloride shows 1000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites. | ||||||||||||||||||||
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RS-127445 hydrochloride (Standard) | 98.56% | RS-127445 (hydrochloride) (Standard) is the analytical standard of RS-127445 (hydrochloride). This product is intended for research and analytical applications. RS-127445 hydrochloride is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. RS-127445 hydrochloride shows 1000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites. | ||||||||||||||||||||
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References
