863115-70-2
863115-70-2
Chemical Structure
MCHR1 antagonist 2
- CAS No.: 863115-70-2
- Formula:C23H21FN2O5
- Molecular Weight:424.42
IUPAC Name: N-(1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)-6-fluoro-4-oxo-4H-chromene-2-carboxamide
InChIKey: HHCYCBKPWYJVEB-UHFFFAOYSA-N
SMILES: O=C(C1=CC(C2=CC(F)=CC=C2O1)=O)NC3CCN(CC4=CC=C(OCO5)C5=C4)CC3
Biological Activity: MCHR1 antagonist 2 is an antagonist of melanin concentrating hormone receptor 1, with an IC50 of 65 nM; MCHR1 antagonist 2 also inhibits hERG, with an IC50 of 4.0 nM in IMR-32 cells[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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MCHR1 antagonist 2 | 98.27% | MCHR1 antagonist 2 is an antagonist of melanin concentrating hormone receptor 1, with an IC50 of 65 nM; MCHR1 antagonist 2 also inhibits hERG, with an IC50 of 4.0 nM in IMR-32 cells. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.57
HY-181861AChE/MAO-B-IN-9 -
Similarity Score 0.53
HY-126130LysRs-IN-2 -
Similarity Score 0.52
HY-B1124AFipexide hydrochloride -
Similarity Score 0.51
HY-B1124RFipexide (Standard) -
Similarity Score 0.51
HY-155999MoTPS1-IN-1 -
Similarity Score 0.51
HY-102089Fluoroclebopride -
Similarity Score 0.50
HY-U00292AMPK activator 1 -
Similarity Score 0.50
HY-160156SSTR5 antagonist 4 -
Similarity Score 0.49
HY-149331TNF-α-IN-11 -
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