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Cat. No.: HY-110054

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CCG-2046

CCG-2046 is a RGS4 inhibitor with an IC₅₀ of 4.3 μM against RGS4-Gα_o interaction signal.

For research use only. We do not sell to patients.

CAS No.: 13017-69-1
Formula: C₁₁H₁₀N₄
Molecular Weight:198.22

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (268 KB)

CCG-2046 Chemical Structure

CAS No.: 13017-69-1

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Bioz

Biological Activity

Description

CCG-2046 is a RGS4 inhibitor with an IC₅₀ of 4.3 μM against RGS4-Gα_o interaction signal^[1].

IC₅₀ & Target

RGS4

4.3 μM (IC₅₀)

All RGS Protein Isoforms :

Chemical Information

CAS No. 13017-69-1
Molecular Weight 198.22
Formula C₁₁H₁₀N₄
SMILES

N#CC1(C(C#N)(C#N)C1(C)CCC)C#N
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (268 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Roman DL, et al. Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay. Mol Pharmacol. 2007 Jan;71(1):169-75. [Content Brief]

Calculators

Molarity Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Dilution Calculator

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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