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Cat. No.: HY-182715

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PSB-10211

PSB-10211 is a P2X2 receptor antagonist with an IC₅₀ of 0.086 μM against rat P2X2 receptors. PSB-10211 inhibits ATP-mediated currents of rat P2X2 receptors expressed in Xenopus oocytes. PSB-10211 can be used in studies related to pain and urinary incontinence.

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CAS No.: 66295-57-6
Formule: C₂₃H₁₃Cl₂N₆NaO₅S
Masse moléculaire:579.35

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Please store the product under the recommended conditions in the Certificate of Analysis.

PSB-10211 Chemical Structure

CAS No.: 66295-57-6

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Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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Activité biologique

Description

Voir tous les produits spécifiques à Isoform P2X Receptor :

In Vitro

PSB-10211 inhibits human P2Y₂ receptor-mediated calcium mobilization with an IC₅₀ of 24.3 μM, shows inhibitory activity with an IC₅₀ of ~10 μM at human P2Y₄ receptors, and shows inhibitory activity at concentrations >10 μM at rat P2Y₆ receptors^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 66295-57-6
Masse moléculaire 579.35
Formule C₂₃H₁₃Cl₂N₆NaO₅S
SMILES

O=C1C2=C(C(C3=C(C(S(=O)(O[Na])=O)=CC(NC4=CC(NC5=NC(Cl)=NC(Cl)=N5)=CC=C4)=C13)N)=O)C=CC=C2
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. Baqi Y, et al. Discovery of potent competitive antagonists and positive modulators of the P2X2 receptor. J Med Chem. 2011;54(3):817-830. [Content Brief]

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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PSB-10211

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Voir tous les produits spécifiques à Isoform P2X Receptor

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PSB-10211 Related Classifications

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