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Cat. No.: HY-103294

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R892

R892 is a selective and efficient bradyK_inin B1 receptor antagonist with significant antagonistic activity. The pA2 values of R892 in human and rabbit B1 receptors are 8.8 and 8.6 respectively, indicating its strong anti-activity at these receptors. R892 exhibits selectivity with ID50 values of 2.8 nM and >600 nM for B1 and B2 receptors, respectively, and has no endogenous agonist activity. R892 is resistant to aminopeptidase and kininase II (ACE) degradation and exhibits metabolic stability.

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CAS No.: 229030-05-1
Formule: C₅₈H₈₃N₁₃O₁₂
Masse moléculaire:1154.36

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Please store the product under the recommended conditions in the Certificate of Analysis.

R892 Chemical Structure

CAS No.: 229030-05-1

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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Description

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Chemical Information

CAS No. 229030-05-1
Masse moléculaire 1154.36
Formule C₅₈H₈₃N₁₃O₁₂
Sequence

Ac-Lys-Arg-Pro-Pro-Gly-{Phe}-Ser-{d-Nal}-Ile
Sequence Shortening

Ac-KRPPG-{Phe}-SA-{d-Nal}-I
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (257 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Kinin B1 receptor antagonists containing alpha-methyl-L-phenylalanine: in vitro and in vivo antagonistic activities

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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R892

Voir tous les produits spécifiques à Isoform Endogenous Metabolite

Activité biologique

Description

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

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HY-103294 Related Classifications

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