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CP-615003

(Synonyms: NGD-913)

CP-615003 is a potent and subtype-selective partial agonist of GABAA receptor (GABAA receptor) (Ki = 1.1 μM). CP-615003 is mainly converted into the active metabolite CP-900725 through oxidative deamination in monkeys and humans, and the latter also has GABAA receptor affinity. CP-615003 is a substrate of P-glycoprotein (P-gp/MDR1), resulting in severe limitation of its penetration into the central nervous system (CNS). CP-615003 can be used for the study of CNS-related indications.

For research use only. We do not sell to patients.

  • CAS No.: 329016-45-7
  • Formula: C20H24FN3O3
  • Molecular Weight:373.42
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • CP-615003 Chemical Structure
    CP-615003 Chemical Structure
CAS No.: 329016-45-7
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  • CP-615003 Chemical Structure
    CP-615003 Chemical Structure
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  • CP-615003