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Cat. No.: HY-W743727

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Cytisine-d₄

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Cytisine-d₄ is the deuterium labeled Cytisinicline (HY-N0175). Cytisinicline (Cytisine) is an alkaloid. Cytisinicline (Cytisine) is a partial agonist of α4β2 nAChRs, and partial to full agonist at β4 containing receptors and α7 receptors. Has been used medically to help with smoking cessation.

For research use only. We do not sell to patients.

CAS No.: 2714473-76-2
Formula: C₁₁H₁₀D₄N₂O
Molecular Weight:194.27

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (248 KB)

Cytisine-d₄ Chemical Structure

CAS No.: 2714473-76-2

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- In Vitro
- Application
Chemical Information
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Biological Activity

Description

Cytisine-d₄ is the deuterium labeled Cytisinicline (HY-N0175). Cytisinicline (Cytisine) is an alkaloid. Cytisinicline (Cytisine) is a partial agonist of α4β2 nAChRs^[1], and partial to full agonist at β4 containing receptors and α7 receptors^[2]. Has been used medically to help with smoking cessation^[3].

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Application

1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.

Chemical Information

CAS No. 2714473-76-2
Unlabeled Cas 485-35-8
Molecular Weight 194.27
Formula C₁₁H₁₀D₄N₂O
SMILES

O=C1N2C[C@@]3(C([2H])(NC([2H])([C@]([H])(C2=CC=C1)C3)[2H])[2H])[H]
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.