D3R/MOR antagonist 1
D3R/MOR antagonist 1 (Compound 114) is a D3R/MOR antagonist (Ki: 46.5 nM and 691 nM respectively). D3R/MOR antagonist 1 has the potential to produce analgesic effects through MOR partial agonism, reduce opioid-misuse liability via D3R antagonism.
For research use only. We do not sell to patients.
- CAS No.: 3033883-15-4
- Formula: C22H27Cl2N3O
- Molecular Weight:420.38
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
46.5 nM and 691 nM (D3R/MOR)[1]
Chemical Information
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CAS No. 3033883-15-4
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Molecular Weight 420.38
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Formula C22H27Cl2N3O
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SMILES
ClC1=C(N2CCN(CCC3(C4=NC=CC=C4)CCOCC3)CC2)C=CC=C1Cl
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)