PSB-CB-27
PSB-CB-27 is a potent and selective GPR18 inhibitor with an IC50 of 0.65 μM. PSB-CB-27 shows selectivity over Human GPR55, Human CB1 receptor, and Human CB2 receptor. PSB-CB-27 leads to a complete blockade of Δ9-Tetrahydrocannabinol (THC)-induced GPR18 activation. PSB-CB-27 can be used for inflammatory diseases and cancer immunotherapy research.
For research use only. We do not sell to patients.
- CAS No.: 2237222-16-9
- Formula: C25H27ClN2O3S
- Molecular Weight:471.01
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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GPR18 0.62 μM (IC50) |
Chemical Information
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CAS No. 2237222-16-9
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Molecular Weight 471.01
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Formula C25H27ClN2O3S
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SMILES
O=C1N2C(SCCC2)=N/C1=C\C3=CC(OCCCCCCOC4=CC=C(C=C4)Cl)=CC=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)