1. Metabolic Enzyme/Protease
    Neuronal Signaling
    GPCR/G Protein
    Membrane Transporter/Ion Channel
  2. Dipeptidyl Peptidase
    GPR119
    Potassium Channel
  3. DPP-4/GPR119 modulator 1

DPP-4/GPR119 modulator 1 

Cat. No.: HY-146468
Handling Instructions

DPP-4/GPR119 modulator 1 (Compound 22) is an orally active dipeptidyl peptidase IV (DPP-IV) inhibitor and GPR119 agonist. DPP-4/GPR119 modulator 1 shows blood glucose-lowering effect and moderate inhibition on hERG channel with an IC50 of 4.9 µM. DPP-4/GPR119 modulator 1 can be used for diabetes research.

For research use only. We do not sell to patients.

DPP-4/GPR119 modulator 1 Chemical Structure

DPP-4/GPR119 modulator 1 Chemical Structure

CAS No. : 2411099-68-6

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Description

DPP-4/GPR119 modulator 1 (Compound 22) is an orally active dipeptidyl peptidase IV (DPP-IV) inhibitor and GPR119 agonist. DPP-4/GPR119 modulator 1 shows blood glucose-lowering effect and moderate inhibition on hERG channel with an IC50 of 4.9 µM. DPP-4/GPR119 modulator 1 can be used for diabetes research[1][1].

IC50 & Target

IC50: 4.9 µM (hERG)[1]

Molecular Weight

623.15

Formula

C30H39ClN10O3

CAS No.
SMILES

CC#CCN1C(N2CCC[[email protected]](C2)N)=NC3=C1C(N(C(N3C)=O)CCCN4CCN(CC4)C5=NC(C6=CC=CC=C6)=NO5)=O.Cl

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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DPP-4/GPR119 modulator 1
Cat. No.:
HY-146468
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