Dyrk1A/B-IN-1
Dyrk1A/B-IN-1 (compound 3n) is a potent, selective and cell-permeable DYRK1A and DYRK1B inhibitor with Kis of 67.8 nM and 237.9 nM, and IC50s of 1.1 μM and 0.8 μM, respectively. Dyrk1A/B-IN-1 is not toxic to human cells. Dyrk1A/B-IN-1 can be used for researching DYRK1A and DYRK1B cellular functions and their role in pathologies.
For research use only. We do not sell to patients.
- CAS No.: 3032401-50-3
- Formula: C21H17N3O2S2
- Molecular Weight:407.51
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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DYRK1A 67.8 nM (Ki) |
DYRK1B 237.9 nM (Ki) |
Chemical Information
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CAS No. 3032401-50-3
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Molecular Weight 407.51
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Formula C21H17N3O2S2
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SMILES
NC(C1=CC2=C(C=CC=C2S1)C3=CC=C(S3)C(NCC4=C(C=CC=C4)N)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Dyrk1A/B-IN-1 Related Classifications
HY-146337 Related Classifications
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