1. GPCR/G Protein
    Neuronal Signaling
  2. Adenosine Receptor
    Monoamine Oxidase
  3. (E)-8-(3-Chlorostyryl)caffeine

(E)-8-(3-Chlorostyryl)caffeine 

Cat. No.: HY-103164
Handling Instructions

(E)-8-(3-Chlorostyryl)caffeine is a selective adenosine A2A receptor antagonist. (E)-8-(3-Chlorostyryl)caffeine inhibits monoamine oxidase B (MAO-B) with a Ki value of 70 nM by a pathway that is independent of its actions on the A2A receptor. (E)-8-(3-Chlorostyryl)caffeine has the potential for Parkinson's disease research.

For research use only. We do not sell to patients.

(E)-8-(3-Chlorostyryl)caffeine Chemical Structure

(E)-8-(3-Chlorostyryl)caffeine Chemical Structure

CAS No. : 147700-11-6

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Description

(E)-8-(3-Chlorostyryl)caffeine is a selective adenosine A2A receptor antagonist. (E)-8-(3-Chlorostyryl)caffeine inhibits monoamine oxidase B (MAO-B) with a Ki value of 70 nM by a pathway that is independent of its actions on the A2A receptor. (E)-8-(3-Chlorostyryl)caffeine has the potential for Parkinson's disease research[1].

IC50 & Target[1]

A2AR

 

MAO-B

70 nM (Ki)

Molecular Weight

330.77

Formula

C16H15ClN4O2

CAS No.
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(E)-8-(3-Chlorostyryl)caffeine
Cat. No.:
HY-103164
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