ASPER-29
ASPER-29 is Asperphenamate HY-129578 analog. ASPER-29 also is a dual cathepsin L and S inhibitor with IC50 value of 6.03 μM and 5.02 μM, respectively. ASPER-29 can be used for the research of the migration and invasion of cancer.
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- No. CAS: 2630388-03-1
- Fòrmula: C31H29BrN2O5S
- Peso molecular:621.54
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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cathepsin L 6.03 μM (IC50) |
cathepsin S 5.02 μM (IC50) |
ASPER-29 has dual Cat L and S inhibitory potency with IC50 value of 6.03 μM and 5.02 μM, respectively[1].
ASPER-29 shows a definite antimetastatic effect on pancreatic cancer BxPC-3 and PANC-1 cells[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 2630388-03-1
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Peso molecular 621.54
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Fòrmula C31H29BrN2O5S
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SMILES
O=C(C1=CC=CC=C1)N[C@@H](C(OC[C@H](NS(=O)(C2=CC=C(C=C2)Br)=O)CC3=CC=CC=C3)=O)CC4=CC=CC=C4
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)