Axelopran
Axelopran (TD-1211) is an opioid receptor antagonist with pKi values of 9.8, 8.8 and 9.9 for human recombinant μ and δ receptors and guinea pig κ receptor, respectively.
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- No. CAS: 949904-48-7
- Fòrmula: C26H39N3O4
- Peso molecular:457.61
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Ver todos los productos específicos de isoformas Opioid Receptor
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Actividad biológica
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guinea pig κ-opioid receptor 9.9 (pKi) |
human μ-opioid receptor 9.8 (pKi) |
δ Opioid Receptor/DOR 8.8 (pKi) |
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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No. CAS 949904-48-7
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Peso molecular 457.61
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Fòrmula C26H39N3O4
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SMILES
O=C([C@@H](O)CO)N(CC1CCCCC1)CCN2[C@H]3C[C@H](C4=CC(C(N)=O)=CC=C4)C[C@@H]2CC3
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Synonyms
TD-1211
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)