DNMT3A-IN-4
DNMT3A-IN-4 is a DNMT3A inhibitor with an IC50 of 33.4 μM against human DNMT3A. DNMT3A-IN-4 inhibits the proliferation of colorectal cancer cells and can be used for the research of colorectal cancer.
Para uso exclusivo en investigación. No vendemos a pacientes.
- Fòrmula: C20H15N5O3
- Peso molecular:373.36
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Actividad biológica
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Chemical Information
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- Pureza y Documentación
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Help & FAQs
Ver todos los productos específicos de isoformas DNA Methyltransferase
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Actividad biológica
Descripciòn
IC50 & Target
[1]|
DNMT3A 33.4 μM (IC50) |
In Vitro
DNMT3A-IN-4 (compound 6o) (100-320 μM; 1 h) preferentially inhibits recombinant human DNMT3A/3L over DNMT1, and shows only weak inhibitory activity against DNMT1 even at concentrations as high as 320 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Peso molecular 373.36
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Fòrmula C20H15N5O3
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SMILES
O=C1NC2=C(C(C3=CC=C(N4C=CN=C4)C=C3)C5=C(O2)C=C(O)C=C5)C(N)=N1
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
DNMT3A-IN-4 Related Classifications
HY-184332 Related Classifications
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