HD-800
HD-800 is a tubulin inhibitor with an IC50 of 4.3 nM and an EC50 for depolymerization of 24 nM. HD-800 can be used to generate a radioactive tracer [11C]HD-800, and [11C]HD-800 can penetrate the blood-brain barrier and be used for positron emission tomography (PET) in various neurological diseases.
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- No. CAS: 1204408-27-4
- Fòrmula: C15H15N3O2
- Peso molecular:269.30
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| 786-0 | GI50 |
10 nM
Compound: 3
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Cytotoxicity against human 786-0 cells assessed as growth inhibition after 48 hrs by SRB assay
Cytotoxicity against human 786-0 cells assessed as growth inhibition after 48 hrs by SRB assay
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[PMID: 27213719] |
Chemical Information
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No. CAS 1204408-27-4
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Peso molecular 269.30
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Fòrmula C15H15N3O2
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SMILES
N=1C=NC(=C2C1OC=C2C)N(C3=CC=C(OC)C=C3)C
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
HD-800 Related Classifications
HY-180347 Related Classifications
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