TM471-1
TM471-1 is an orally active and covalent Bruton's tyrosine kinase (BTK) inhibitor with IC50 values of 1.3 nM (BTKWT), >40,000 nM (BTKC481S), 7.9 nM (TEC) and 12.4 nM (TXK). TM471-1 inhibits cell growth in vivo and in vitro, arrests cell cycle at G0/G1 phase and induces cell apoptosis.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 2649008-95-5
- Fòrmula: C27H29N5O3
- Peso molecular:471.55
-
Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Actividad biológica
-
Chemical Information
- Pureza y Documentación
- Referencias
-
Help & FAQs
Actividad biológica
Chemical Information
-
No. CAS 2649008-95-5
-
Peso molecular 471.55
-
Fòrmula C27H29N5O3
-
SMILES
O=C(N)C1=C(C2=CC=C(OC3=CC=CC=C3)C=C2)N=C4N1NCC[C@H]4C5CCN(C(C=C)=O)CC5
-
Envío
Room temperature in continental US; may vary elsewhere.
-
Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
TM471-1 Related Classifications
HY-174129 Related Classifications
Powered by Bioz