TP-680
TP-680 is a cholecystokinin receptor antagonist. TP-680 binds 1510 times more strongly to rat pancreatic CCKA receptors (IC50=1.2 nM) than to rat brain CCKB receptors (IC50=1812.5 nM). TP-680 can be used in the study of gastrointestinal diseases.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 176915-07-4
- Fòrmula: C35H33N5O4S
- Peso molecular:619.73
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
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CCKAR 1.2 nM (IC50) |
CCKBR 1812.5 nM (IC50) |
Chemical Information
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No. CAS 176915-07-4
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Peso molecular 619.73
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Fòrmula C35H33N5O4S
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SMILES
O=C(O)C1=CC=CN=C1SC[C@@H](C(N2CCN(CC2)C(C3=CC=CC=C3)C4=CC=CC=C4)=O)NC(C5=CC6=C(C=CC=C6)N5)=O
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)