2. Metabolic Enzyme/Protease
  3. Phospholipase
  4. Giripladib

Giripladib (PLA-695) is a indole-based inhibitor of cytosolic phospholipase A2 (cPLA2). Giripladib can be used for osteoarthritis and breast cancer research.

For research use only. We do not sell to patients.

Giripladib Chemical Structure

Giripladib Chemical Structure

CAS No. : 865200-20-0

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Based on 1 publication(s) in Google Scholar

Giripladib Related Antibodies

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Description

Giripladib (PLA-695) is a indole-based inhibitor of cytosolic phospholipase A2 (cPLA2). Giripladib can be used for osteoarthritis and breast cancer research[1][2].

IC50 & Target

cPLA2α

 

Clinical Trial
Molecular Weight

745.25

Formula

C41H36ClF3N2O4S
CAS No.
Appearance

Solid

Color

White to light yellow

SMILES

O=C(C1=CC=C(CCCC2=C(CCNS(=O)(CC3=C(C(F)(F)F)C=CC=C3)=O)N(C(C4=CC=CC=C4)C5=CC=CC=C5)C6=C2C=C(C=C6)Cl)C=C1)O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
Purity & Documentation
References
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Giripladib Related Classifications

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Giripladib865200-20-0PLA-695PLA695PLA 695PhospholipaseOsteoarthritisBCSCstumorigenesisbreast cancer stem cellscytosolic phospholipase A2Inhibitorinhibitorinhibit

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