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Cat. No.: HY-186385

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GPR39 antagonist-2

GPR39 antagonist-2 is a GPR39 antagonist. GPR39 antagonist-2 is used in research on various diseases such as cardiovascular diseases, endocrine system and hormonal disorders, cancer, and metabolic diseases.

For research use only. We do not sell to patients.

CAS No.: 2924750-68-3
Formula: C₂₁H₂₄F₂N₆O
Molecular Weight:414.45

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

GPR39 antagonist-2 Chemical Structure

CAS No.: 2924750-68-3

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- In Vitro
Chemical Information
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Biological Activity

Description

In Vitro

GPR39 antagonist-2 (Compound 51) modulates calcium responses in PC3 cells expressing endogenous GPR39 receptors, with an fpKi of ≥ 7.3^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 2924750-68-3
Molecular Weight 414.45
Formula C₂₁H₂₄F₂N₆O
SMILES

O=C(N1CCC(F)(CC1)F)C2=C(C3=NN(C(C)C)C=C3)C=C(C4=NN=C(C)N4)C=C2
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Agostino CIANCIULLI, et al. Antagonists of gpr39 protein. WO2023076219A2. WIPO (PCT). 2022-10-25.

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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