GPR55 agonist 3
Based on 1 Customer Validation
GPR55 agonist 3 (Compound 26) is a GPR55 agonist (EC50: 0.239 nM, and 1.76 nM for hGPR55 and rGPR55). GPR55 agonist 3 induces β-arrestin recruitment to human GPR55 (EC50: 6.2 nM).
For research use only. We do not sell to patients.
- Purity: 99.17%
- CAS No.: 3006105-44-5
- Formula: C19H16F4N4
- Molecular Weight:376.35
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
Biological Activity
Chemical Information
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CAS No. 3006105-44-5
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Appearance Solid
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Molecular Weight 376.35
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Formula C19H16F4N4
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Color White to off-white
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SMILES
FC(F)(F)CC1=CN=CC(C2=CN=C(N[C@@H](C3=CC=C(F)C=C3)C)C=N2)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 250 mg/mL (664.28 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (266 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.6571 mL | 13.2855 mL | 26.5710 mL | 66.4275 mL |
| 5 mM | 0.5314 mL | 2.6571 mL | 5.3142 mL | 13.2855 mL | |
| 10 mM | 0.2657 mL | 1.3286 mL | 2.6571 mL | 6.6428 mL | |
| 15 mM | 0.1771 mL | 0.8857 mL | 1.7714 mL | 4.4285 mL | |
| 20 mM | 0.1329 mL | 0.6643 mL | 1.3286 mL | 3.3214 mL | |
| 25 mM | 0.1063 mL | 0.5314 mL | 1.0628 mL | 2.6571 mL | |
| 30 mM | 0.0886 mL | 0.4429 mL | 0.8857 mL | 2.2143 mL | |
| 40 mM | 0.0664 mL | 0.3321 mL | 0.6643 mL | 1.6607 mL | |
| 50 mM | 0.0531 mL | 0.2657 mL | 0.5314 mL | 1.3286 mL | |
| 60 mM | 0.0443 mL | 0.2214 mL | 0.4429 mL | 1.1071 mL | |
| 80 mM | 0.0332 mL | 0.1661 mL | 0.3321 mL | 0.8303 mL | |
| 100 mM | 0.0266 mL | 0.1329 mL | 0.2657 mL | 0.6643 mL |