GPR84 agonist-2
Based on 1 Customer Validation
GPR84 agonist-2 is a selective GPR84 agonist with no activity at free fatty acid receptors. GPR84 agonist-2 enhances GPR84-mediated signaling above basal levels and potentiates agonist-induced GPR84 activation. GPR84 agonist‑2 can be used for research on GPR84-related physiological mechanisms.
For research use only. We do not sell to patients.
- Purity: 99.80%
- CAS No.: 3105662-82-3
- Formula: C21H35NO2
- Molecular Weight:333.51
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Storage:
4°C, stored under nitrogen
* In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
Biological Activity
GPR84 agonist‑2 (compound 8e) acts as a full agonist at human GPR84 with a pEC50 of 6.24 and 100% efficacy, and exhibits no inverse agonistic or antagonistic activity in the PRESTO‑Tango β‑arrestin recruitment assay[1].
GPR84 agonist-2 are selective, showing no significant activity on related free fatty acid receptors FFA1, FFA2, FFA3, or FFA4[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3105662-82-3
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Appearance Oil
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Molecular Weight 333.51
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Formula C21H35NO2
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Color Yellow to brown
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SMILES
OC1=CC(OCC2CCCCC2)=NC(CCCCCCCCC)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
4°C, stored under nitrogen
* In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
Purity & Documentation
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Data Sheet (263 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)