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Cat. No.: HY-116554

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GYKI-46903

GYKI-46903 is a non-competitive antagonist for 5-HT3 receptor, with the pIC₅₀ of 6.91.

For research use only. We do not sell to patients.

CAS No.: 142999-59-5
Formula: C₁₇H₂₁ClFNO₂
Molecular Weight:325.81

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (268 KB)

GYKI-46903 Chemical Structure

CAS No.: 142999-59-5

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

GYKI-46903 is a non-competitive antagonist for 5-HT3 receptor, with the pIC₅₀ of 6.91^[1].

All 5-HT Receptor Isoforms :

Chemical Information

CAS No. 142999-59-5
Molecular Weight 325.81
Formula C₁₇H₂₁ClFNO₂
SMILES

CCC(O[C@H]1[C@@]2([H])C(C3=CC=C(C=C3)F)=CC[N@@](CC1)C2)=O.Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (268 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. V Csillik-Perczel, et al. GYKI-46 903, a Non-Competitive Antagonist for 5-HT3 Receptors. Comparative Study Pharmacol Toxicol. 1996 Jul;79(1):32-9. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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