HSR-IN-1
HSR-IN-1 (Compound 28) is an effective hSR (human serine racemase) inhibitor. In the presence of the cofactor Pyridoxal 5'-phosphate monohydrate (HY-W011727A), HSR-IN-1 has a Kd value of 5.4 μM and an IC50 of 18.3 μM for hSR, while the IC50 of HSR-IN-1 alone is 4.7 μM. HSR-IN-1 can be used for research on central nervous system diseases.
For research use only. We do not sell to patients.
- Formula: C15H16ClNO3
- Molecular Weight:293.75
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 4.7 μM (Human Serine Racemase (HSR))
HSR-IN-1 (2-150 μM, 5 min) tightly binds to hSR and exhibits strong inhibitory activity against hSR activity[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 293.75
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Formula C15H16ClNO3
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SMILES
[NH3+]OC(C(O)=O)CC1=CC=C(C2=CC=CC=C2)C=C1.[Cl-]
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)