HSR-IN-1
HSR-IN-1 (Compound 28) is an effective hSR (human serine racemase) inhibitor. In the presence of the cofactor Pyridoxal 5'-phosphate monohydrate (HY-W011727A), HSR-IN-1 has a Kd value of 5.4 μM and an IC50 of 18.3 μM for hSR, while the IC50 of HSR-IN-1 alone is 4.7 μM. HSR-IN-1 can be used for research on central nervous system diseases.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- Formel: C15H16ClNO3
- Molecular Weight:293.75
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
Beschreibung
IC50 & Target
IC50: 4.7 μM (Human Serine Racemase (HSR))
In Vitro
HSR-IN-1 (2-150 μM, 5 min) tightly binds to hSR and exhibits strong inhibitory activity against hSR activity[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 293.75
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Formel C15H16ClNO3
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SMILES
[NH3+]OC(C(O)=O)CC1=CC=C(C2=CC=CC=C2)C=C1.[Cl-]
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)