Hit 1
Hit 1 is an activator of ansulin degrading enzyme (IDE), with an EC50 of 5.5 μM. Hit 1 can decrease glucose-stimulating insulin secretion.
For research use only. We do not sell to patients.
- CAS No.: 2785377-42-4
- Formula: C22H24N4O3S2
- Molecular Weight:456.58
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
EC50: 5.5 μM (ansulin degrading enzyme)[1]
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 2785377-42-4
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Molecular Weight 456.58
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Formula C22H24N4O3S2
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SMILES
O=C(NCCCN1C=CN=C1)CCCC2=CN(C3=CC=CC=C23)S(=O)(C4=CC=CS4)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)