SA72
SA72 is a highly selective fatty acid amide hydrolase (FAAH) inhibitor.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 934809-60-6
- 分子式: C21H26N2O6
- 分子量:402.44
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
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HY-14380
PF-3845FAAH Inhibitor -
HY-14376
RedafamdastatFAAH Inhibitor -
HY-N2365
Macamide BFAAH Inhibitor -
HY-10865
LY2183240Anandamide Uptake/FAAH Inhibitor -
HY-19740
BIA 10-2474FAAH Inhibitor -
HY-79511
FAAH-IN-2FAAH Inhibitor -
HY-10862
FAAH inhibitor 1FAAH Inhibitor -
HY-19636
JNJ-42165279FAAH Inhibitor -
HY-10864
URB-597FAAH Inhibitor -
HY-79511R
FAAH-IN-2 (Standard)FAAH Inhibitor -
HY-14376R
Redafamdastat (Standard)FAAH Inhibitor -
HY-N2365R
Macamide B (Standard)FAAH Inhibitor
生物活性
製品説明
IC50 & Target
Fatty acid amide hydrolase (FAAH)[1]
体外実験
Fatty acid amide hydrolase (FAAH) is the primary regulator of several bioactive lipid amides including anandamide. Inhibitors of FAAH are potentially useful for the treatment of pain, anxiety, depression, and other nervous system disorders. However, FAAH inhibitors must display selectivity for this enzyme relative to the numerous other serine hydrolases present in the human proteome in order to be therapeutically acceptable. SA-72 is also a carbamate inhibitor. However, SA-72 shows exceptional selectivity for FAAH. Tested carboxylesterases are not off-targets for SA-72. SA-72 does not have major effects on the level of carboxylesterase activities in liver microsomes[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .
化学情報
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CAS 番号 934809-60-6
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分子量 402.44
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分子式 C21H26N2O6
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SMILES
O=C(OCC(N)=O)NCCCC1OCC(C2=C3C=CC(OC)=CC3=CC=C2)CO1
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
SA72 関連分類
HY-U00240 関連分類
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