country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Country or Region:

United States

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

製品番号: HY-107723A

Copy Link Print Information

CGP71683

CGP 71683 Free base serves as a powerful and highly selective non-peptide antagonist targeting the NPY Y(5) receptor, making it a valuable tool in obesity research.

商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。

CAS 番号: 192321-23-6
分子式: C₂₆H₂₉N₅O₂S
分子量:475.61

保管条件:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (241 KB)

CGP71683 構造式

CAS 番号: 192321-23-6

容量

価格（税別）

在庫状況

数量

Amount: USD 0.00

* アイテムを追加する前、数量をご選択ください

Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

生物活性

製品説明

CGP 71683 Free base serves as a powerful and highly selective non-peptide antagonist targeting the NPY Y(5) receptor, making it a valuable tool in obesity research.

Neuropeptide Y Receptor アイソフォーム固有の製品をすべて表示 :

Cellular Effect

Cell Line	Type	Value	Description	References
COS-1	IC₅₀	1.3 nM Compound: CGP-71683A (Trans)	Inhibitory activity against constitutively activated human Neuropeptide Y receptor Y5 transiently expressed in COS-1 cells using [125I]PYY Inhibitory activity against constitutively activated human Neuropeptide Y receptor Y5 transiently expressed in COS-1 cells using [125I]PYY	[PMID: 15863317]
COS-1	IC₅₀	97 nM Compound: CGP-71683A (Trans)	Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]MK-912 Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]MK-912	[PMID: 15863317]
HEK293	IC₅₀	3500 nM Compound: CGP-71683A (Trans)	Inhibitory activity against mutated constitutively activated human Melanin concentrating hormone receptor 1 (CA-MCH-R1) stably expressed in HEK293 cells using [125I](Phe13, Tyr19) MCH Inhibitory activity against mutated constitutively activated human Melanin concentrating hormone receptor 1 (CA-MCH-R1) stably expressed in HEK293 cells using [125I](Phe13, Tyr19) MCH	[PMID: 15863317]

化学情報

CAS 番号 192321-23-6
分子量 475.61
分子式 C₂₆H₂₉N₅O₂S
SMILES

NC1=NC(NC[C@@H](CC2)CC[C@H]2CNS(=O)(C3=CC=CC4=CC=CC=C34)=O)=NC5=CC=CC=C51
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

Please store the product under the recommended conditions in the Certificate of Analysis.