Pumosetrag
Based on 1 publication(s) in Google Scholar
Pumosetrag is a bioavtive small molecular compound.
연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.
- CAS No.: 153062-94-3
- 화학식: C15H17N3O2S
- 분자량:303.38
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications Citing Use of MedChemExpress (MCE) Pumosetrag
MoreAll 5-HT Receptor Isoforms
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Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HEK293 | EC50 |
5.4 nM
Compound: DDP733
|
Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced response
Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced response
|
[PMID: 21146988] |
| HEK293 | EC50 |
9.2 nM
Compound: DDP733
|
Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as decrease in 10 uM 5-chloroindole-induced increase in intracellular calcium release
Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as decrease in 10 uM 5-chloroindole-induced increase in intracellular calcium release
|
[PMID: 21146988] |
Chemical Information
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CAS No. 153062-94-3
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분자량 303.38
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화학식 C15H17N3O2S
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SMILES
O=C(C1=CNC(C=CS2)=C2C1=O)N[C@@H]3C4CCN(CC4)C3
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications (1)
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Journal Impact Factor
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Most Recent
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Expert Opin Pharmacother
Recent advances in the pharmacological management of constipation predominant irritable bowel syndrome. [Abstract]2020 Jan;21(1):73-84. PMID: 31724881
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)