2. Metabolic Enzyme/Protease
  3. Stearoyl-CoA Desaturase (SCD)
  4. MK-8245 analog

MK-8245 analog (compound 6) is a potent stearoyl-CoA desaturase (SCD) inhibitor with an IC50 of 7 nM for rat SCD. MK-8245 analog has antidiabetic and antidyslipidemic effects.

For research use only. We do not sell to patients.

MK-8245 analog Chemical Structure

MK-8245 analog Chemical Structure

CAS No. : 1030612-87-3

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MK-8245 analog Related Antibodies

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Description

MK-8245 analog (compound 6) is a potent stearoyl-CoA desaturase (SCD) inhibitor with an IC50 of 7 nM for rat SCD. MK-8245 analog has antidiabetic and antidyslipidemic effects[1].

IC50 & Target

IC50: 7 nM (rat SCD)[1]
Molecular Weight

484.30

Formula

C16H15BrFN7O3S
CAS No.
SMILES

O=C(O)CN1N=C(C2=NN=C(N3CCC(OC4=CC(F)=CC=C4Br)CC3)S2)N=N1
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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MK-8245 analog Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MK-82451030612-87-3MK8245MK 8245Stearoyl-CoA Desaturase (SCD)SCD inhibitorantidiabetic and antidyslipidemic effectsInhibitorinhibitorinhibit

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MK-8245 analog
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HY-114184
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